Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL

LigandBDBM50159729(4-[3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]p...)Copy SMILESCopy InChI

Affinity DataKi:  42nMAssay Description:Binding affinity towards Adenosine A2A receptor of rat brain tissues using [3H]-ZM-241,385 as radioligandMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetAdenosine receptor A1(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL

LigandBDBM50159729(4-[3-(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]p...)Copy SMILESCopy InChI

Affinity DataKi:  66nMAssay Description:Binding affinity towards Adenosine A1 receptor of rat cerebral cortex using [3H]-DPCPX as radioligandMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI