Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286749((3S,4S)-3-Pyridin-3-ylmethyl-7-(1-quinolin-2-yl-et...)
Affinity DataKi:  5.20E+3nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50286749((3S,4S)-3-Pyridin-3-ylmethyl-7-(1-quinolin-2-yl-et...)
Affinity DataKi: >5.00E+4nMAssay Description:In vitro inhibitory activity against leukotriene D4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286749((3S,4S)-3-Pyridin-3-ylmethyl-7-(1-quinolin-2-yl-et...)
Affinity DataIC50:  3.80E+4nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4) induced ChemotaxisMore data for this Ligand-Target Pair
In DepthDetails Article