Home
About
Info
Download
WebServices
Contact
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Lysine-specific demethylase 2B
(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Ligand
BDBM319654
(2-[1-(1-phenylethyl)-1H-imidazol-4-yl]-4-[5- (trif...)
Copy SMILES
Affinity Data
IC50: <100nM
Assay Description:
The ability of test compounds to inhibit the activity of FBXL10 was determined in 384-well plate format under the following reaction conditions: 0.3 ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Ligand
BDBM319654
(2-[1-(1-phenylethyl)-1H-imidazol-4-yl]-4-[5- (trif...)
Copy SMILES
Affinity Data
IC50: 300nM
Assay Description:
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384-well plate format under the following reaction conditions: 0.8...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Lysine-specific demethylase 4C
(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Ligand
BDBM319654
(2-[1-(1-phenylethyl)-1H-imidazol-4-yl]-4-[5- (trif...)
Copy SMILES
Affinity Data
IC50: >1.00E+4nM
Assay Description:
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Lysine-specific demethylase 6B
(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Ligand
BDBM319654
(2-[1-(1-phenylethyl)-1H-imidazol-4-yl]-4-[5- (trif...)
Copy SMILES
Affinity Data
IC50: >1.00E+4nM
Assay Description:
The ability of test compounds to inhibit the activity of JMJD3 was determined in 384-well plate format under the following reaction conditions: 1 nM ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI