Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 10 hits in this display
BDBM50388626(CHEMBL2059435 | US9296736, 152 | US9593129, Exampl...)
BDBM50388626(CHEMBL2059435 | US9296736, 152 | US9593129, Exampl...)
BDBM50388626(CHEMBL2059435 | US9296736, 152 | US9593129, Exampl...)
IC50: 1.10nMAssay Description:Binding affinity to human GST-thrombin-tagged MDM2 assessed as inhibition of interaction with human p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
BDBM50388626(CHEMBL2059435 | US9296736, 152 | US9593129, Exampl...)
BDBM50388626(CHEMBL2059435 | US9296736, 152 | US9593129, Exampl...)
BDBM50388626(CHEMBL2059435 | US9296736, 152 | US9593129, Exampl...)
BDBM50388626(CHEMBL2059435 | US9296736, 152 | US9593129, Exampl...)
IC50: 760nMAssay Description:Activity at p53 in human SJSA1 cells assessed as induction of p21 mRNA expression after 7 hrs by qRT-PCR analysis in presence of 10% human serumMore data for this Ligand-Target Pair
BDBM50388626(CHEMBL2059435 | US9296736, 152 | US9593129, Exampl...)
BDBM50388626(CHEMBL2059435 | US9296736, 152 | US9593129, Exampl...)
BDBM50388626(CHEMBL2059435 | US9296736, 152 | US9593129, Exampl...)