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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetNicotinic acetylcholine receptor alpha9/alpha10(RAT)
Hainan University

Curated by ChEMBL
LigandPNGBDBM50445324(CHEMBL3104237)
Affinity DataIC50:  19nMAssay Description:Antagonist activity at Sprague-Dawley rat alpha9alpha10 nAChR expressed in Xenopus oocytes assessed as inhibition of ACh-induced current by voltage c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha9/alpha10(RAT)
Hainan University

Curated by ChEMBL
LigandPNGBDBM50445324(CHEMBL3104237)
Affinity DataIC50:  109nMAssay Description:Inhibition of rat alpha9alpha10 nAChRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-3(Rattus norvegicus)
Hainan University

Curated by ChEMBL
LigandPNGBDBM50445324(CHEMBL3104237)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at Sprague-Dawley rat alpha6/alpha3beta2beta3 nAChR expressed in Xenopus oocytes assessed as inhibition of ACh-induced current by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Hainan University

Curated by ChEMBL
LigandPNGBDBM50445324(CHEMBL3104237)
Affinity DataIC50:  980nMAssay Description:Antagonist activity at Sprague-Dawley rat alpha6/alpha3beta4 nAChR expressed in Xenopus oocytes assessed as inhibition of ACh-induced current by volt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50445324(CHEMBL3104237)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at human alpha9alpha10 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of ACh-induced current amplitude at -80 m...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50445324(CHEMBL3104237)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human alpha9alpha10 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of ACh-evoked currents by two-electrode voltage cl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Hainan University

Curated by ChEMBL
LigandPNGBDBM50445324(CHEMBL3104237)
Affinity DataIC50:  4.20E+3nMAssay Description:Antagonist activity at Sprague-Dawley rat alpha3beta4 nAChR expressed in Xenopus oocytes assessed as inhibition of ACh-induced current by voltage cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50445324(CHEMBL3104237)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of rat alpha7 nAChRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50445324(CHEMBL3104237)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human alpha7 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of ACh-evoked currents by two-electrode voltage clamp ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed