Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetG protein-coupled receptor kinase 5(Homo sapiens (Human))
Universit£

Curated by ChEMBL

LigandBDBM50191326(CHEMBL3953837)Copy SMILESCopy InChI

Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of recombinant human GRK5 expressed in Sf9 insect cells assessed as decrease in phosphorylation of urea-washed bovine rod outer segments i...More data for this Ligand-Target Pair

Target InfoPDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetBeta-adrenergic receptor kinase 2(Bos taurus)
Universit£

Curated by ChEMBL

LigandBDBM50191326(CHEMBL3953837)Copy SMILESCopy InChI

Affinity DataIC50:  2.26E+4nMAssay Description:Inhibition of recombinant bovine GRK3 expressed in Sf9 insect cells assessed as decrease in phosphorylation of urea-washed bovine rod outer segments ...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI