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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Kappa-type opioid receptor
(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50051597
(CHEMBL269119 | Dynorphin A analogues)
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Affinity Data
IC50: 230nM
Assay Description:
Inhibition of binding [3H]U-69,539 at Opioid receptor kappa 1 of guinea pig brain membrane (GPB) homogenates.
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Mu-type opioid receptor
(GUINEA PIG)
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50051597
(CHEMBL269119 | Dynorphin A analogues)
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Affinity Data
IC50: 5.10E+3nM
Assay Description:
Inhibition of binding [3H]-DAMGO at Opioid receptor mu 1 of guinea pig brain membrane (GPB) homogenates.
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Delta-type opioid receptor
(MOUSE)
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50051597
(CHEMBL269119 | Dynorphin A analogues)
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Affinity Data
IC50: >6.00E+4nM
Assay Description:
Agonistic activity towards Opioid receptor delta 1 was determined by evaluating the inhibitory activity towards electrically stimulated mouse vas def...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI