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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
8
hits in this display
Target
Kappa-type opioid receptor
(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by
ChEMBL
Ligand
BDBM50059581
(CHEMBL406893 | N,N-diCPM[D-Pro-10]Dyn A-(1-11))
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Affinity Data
Ki: 0.190nM
Assay Description:
Affinity against Opioid receptor kappa 1 was determined by measuring the inhibition of [3H]-bremazocine binding to guinea pig cerebellar membranes
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Kappa-type opioid receptor
(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by
ChEMBL
Ligand
BDBM50059581
(CHEMBL406893 | N,N-diCPM[D-Pro-10]Dyn A-(1-11))
Copy SMILES
Copy InChI
Affinity Data
Ki: 2.60nM
Assay Description:
Affinity against Opioid receptor kappa 1 was determined by measuring the inhibition of [3H]U69,593 binding to guinea pig cerebellar membranes
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mu-type opioid receptor
(Rattus norvegicus (rat))
Oregon State University
Curated by
ChEMBL
Ligand
BDBM50059581
(CHEMBL406893 | N,N-diCPM[D-Pro-10]Dyn A-(1-11))
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Affinity Data
Ki: 3.90nM
Assay Description:
Affinity against Opioid receptor mu 1 was determined by measuring the inhibition of [3H]-DAMGO binding to rat forebrain membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Kappa-type opioid receptor
(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by
ChEMBL
Ligand
BDBM50059581
(CHEMBL406893 | N,N-diCPM[D-Pro-10]Dyn A-(1-11))
Copy SMILES
Copy InChI
Affinity Data
Ki: 44nM
Assay Description:
Affinity against Opioid receptor kappa 3 was determined by measuring the inhibition of [3H]-NalBzoH binding to guinea pig cerebellar membranes
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Delta-type opioid receptor
(Rattus norvegicus (rat))
Oregon State University
Curated by
ChEMBL
Ligand
BDBM50059581
(CHEMBL406893 | N,N-diCPM[D-Pro-10]Dyn A-(1-11))
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Copy InChI
Affinity Data
Ki: 166nM
Assay Description:
Affinity against Opioid receptor delta 1 was determined by measuring the inhibition of [3H]-DPDPE binding to rat forebrain membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Kappa-type opioid receptor
(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by
ChEMBL
Ligand
BDBM50059581
(CHEMBL406893 | N,N-diCPM[D-Pro-10]Dyn A-(1-11))
Copy SMILES
Copy InChI
Affinity Data
IC50: 3.30nM
Assay Description:
Binding affinity of the compound towards Opioid receptor kappa 1 using [3H]-diprenorphine as radioligand in guinea pig cerebellar membrane in absence...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Kappa-type opioid receptor
(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by
ChEMBL
Ligand
BDBM50059581
(CHEMBL406893 | N,N-diCPM[D-Pro-10]Dyn A-(1-11))
Copy SMILES
Copy InChI
Affinity Data
IC50: 29nM
Assay Description:
Binding affinity of the compound towards Opioid receptor kappa 1 using [3H]-diprenorphine as radioligand in guinea pig cerebellar membrane in presenc...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Kappa-type opioid receptor
(Cavia porcellus (domestic guinea pig))
Oregon State University
Curated by
ChEMBL
Ligand
BDBM50059581
(CHEMBL406893 | N,N-diCPM[D-Pro-10]Dyn A-(1-11))
Copy SMILES
Copy InChI
Affinity Data
IC50: 388nM
Assay Description:
Affinity against Opioid receptor kappa 2 was determined by measuring the inhibition of [3H]-bremazocine binding to guinea pig cerebellar membranes
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI