Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetAminopeptidase N(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50415634(CHEMBL260622)
Affinity DataKi:  100nMAssay Description:Inhibition of catalytic activity of human aminopeptidase N transfected in HEK293 cells assessed as formation of p-nitroanilineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50415634(CHEMBL260622)
Affinity DataKi:  100nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50415634(CHEMBL260622)
Affinity DataKi:  550nMAssay Description:Displacement of [3H]valsartan from human AT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50415634(CHEMBL260622)
Affinity DataKi:  4.46E+3nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50415634(CHEMBL260622)
Affinity DataKi:  4.47E+3nMAssay Description:Inhibition of catalytic activity of human IRAP transfected in HEK293 cells assessed as formation of p-nitroanilineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed