Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAminopeptidase N(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50415636(CHEMBL1077590)
Affinity DataKi:  219nMAssay Description:Inhibition of catalytic activity of human aminopeptidase N transfected in HEK293 cells assessed as formation of p-nitroanilineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50415636(CHEMBL1077590)
Affinity DataKi:  2.45E+3nMAssay Description:Inhibition of catalytic activity of human IRAP transfected in HEK293 cells assessed as formation of p-nitroanilineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed