Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50210542((2S,3S)-methyl 2-(2-((S)-2,6-dioxo-3-(3,4,5-trimet...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of MMP2 after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50210542((2S,3S)-methyl 2-(2-((S)-2,6-dioxo-3-(3,4,5-trimet...)
Affinity DataIC50:  4.93E+4nMAssay Description:Inhibition of pig kidney microsomal aminopeptidase assessed as liberation of p-nitroanilideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50210542((2S,3S)-methyl 2-(2-((S)-2,6-dioxo-3-(3,4,5-trimet...)
Affinity DataIC50:  4.93E+4nMAssay Description:Inhibition of pig kidney microsomes aminopeptidase N preincubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed