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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Kappa-type opioid receptor
(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50038017
(CHEMBL263509 | Tyr-Gly-Gly-Phe-D-Pen-Arg-Arg-Ile-A...)
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Affinity Data
IC50: 71nM
Assay Description:
Binding affinity at kappa opioid receptor in guinea pig brain by [3H]U-69,593 displacement.
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Mu-type opioid receptor
(GUINEA PIG)
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50038017
(CHEMBL263509 | Tyr-Gly-Gly-Phe-D-Pen-Arg-Arg-Ile-A...)
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Affinity Data
IC50: 563nM
Assay Description:
Binding affinity at mu opioid receptor in guinea pig brain by [3H]-DAMGO displacement.
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Delta-type opioid receptor
(Homo sapiens (Human))
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50038017
(CHEMBL263509 | Tyr-Gly-Gly-Phe-D-Pen-Arg-Arg-Ile-A...)
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Copy InChI
Affinity Data
IC50: 1.91E+3nM
Assay Description:
Binding affinity at delta opioid receptor in guinea pig brain by [3H]c[D-Pen2, p-Cl-Phe4, D-Pen5]-enkephalin displacement.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI