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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
8
hits in this display
Target
Melanocortin receptor 4
(Rattus norvegicus)
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50373472
(CHEMBL429854)
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Affinity Data
IC50: 1.70nM
Assay Description:
Binding affinity to rat MC4R
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 4
(Homo sapiens (Human))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50373472
(CHEMBL429854)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4nM
Assay Description:
Displacement of [125I]NDP-alpha-MSH from human MC4R expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 5
(Homo sapiens (Human))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50373472
(CHEMBL429854)
Copy SMILES
Copy InChI
Affinity Data
IC50: 65nM
Assay Description:
Binding affinity to human MC5R
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 3
(Homo sapiens (Human))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50373472
(CHEMBL429854)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.05E+3nM
Assay Description:
Binding affinity to human MC3R
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 5
(Homo sapiens (Human))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50373472
(CHEMBL429854)
Copy SMILES
Copy InChI
Affinity Data
EC50: 102nM
Assay Description:
Agonist activity at human MC5R expressed in CHO cells assesses as cAMP release
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 4
(Rattus norvegicus)
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50373472
(CHEMBL429854)
Copy SMILES
Copy InChI
Affinity Data
EC50: 0.5nM
Assay Description:
Binding affinity to rat MC4R
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 3
(Homo sapiens (Human))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50373472
(CHEMBL429854)
Copy SMILES
Copy InChI
Affinity Data
EC50: 97nM
Assay Description:
Agonist activity at human MC3R expressed in CHO cells assessed as cAMP release
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 4
(Homo sapiens (Human))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50373472
(CHEMBL429854)
Copy SMILES
Copy InChI
Affinity Data
EC50: 2.10nM
Assay Description:
Agonist activity at human MC4R expressed in CHO cells assessed as cAMP release
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI