Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetAndrogen receptor(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154007(11-Ethyl-17-hydroxy-13-methyl-1,2,6,7,8,11,12,13,1...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human androgen receptor expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154007(11-Ethyl-17-hydroxy-13-methyl-1,2,6,7,8,11,12,13,1...)
Affinity DataIC50:  55nMAssay Description:Inhibition of human lymph node carcinoma of prostate (LNCaP) cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154007(11-Ethyl-17-hydroxy-13-methyl-1,2,6,7,8,11,12,13,1...)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibition of CHO-K1 cells expressing glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed