Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetCholinesterase(Equus caballus (Horse))
Martin-Luther-Universit£T Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50175878(4-bromobutyl (4aS,6aS,6bR,8aR,10R,11R,12aR,12bR,14...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 20mins before the addition of substrate by Ellman's met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Martin-Luther-Universit£T Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50175878(4-bromobutyl (4aS,6aS,6bR,8aR,10R,11R,12aR,12bR,14...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate preincubated for 20mins before the addition of substrate by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50175878(4-bromobutyl (4aS,6aS,6bR,8aR,10R,11R,12aR,12bR,14...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 mins by microplate reader bas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50175878(4-bromobutyl (4aS,6aS,6bR,8aR,10R,11R,12aR,12bR,14...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed