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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universita Degli Studi Di Torino

Curated by ChEMBL
LigandPNGBDBM50324377(4-(5-(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphth...)
Affinity DataEC50:  1.50E+3nMAssay Description:Inhibition of MDR1 expressed in MDCK cells assessed as calcein AM accumulation by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Universita Degli Studi Di Torino

Curated by ChEMBL
LigandPNGBDBM50324377(4-(5-(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphth...)
Affinity DataEC50:  2.80E+3nMAssay Description:Inhibition of MRP1 expressed in MDCK cells assessed as calcein AM accumulation by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed