Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetRibosomal protein S6 kinase alpha-5(Homo sapiens (Human))
Astrazeneca R&D Griffith University

Curated by ChEMBL
LigandPNGBDBM50269822(16,25-dihydroxy-13(24),17-cheilanthadien-19,25-oli...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of MSK1 (unknown origin) assessed as [33P] incorporation by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Astrazeneca R&D Griffith University

Curated by ChEMBL
LigandPNGBDBM50269822(16,25-dihydroxy-13(24),17-cheilanthadien-19,25-oli...)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibition of MAPKAPK2 (unknown origin) assessed as [33P] incorporation by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed