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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
72 kDa type IV collagenase
(Homo sapiens (Human))
Abbott Laboratories
Curated by
ChEMBL
Ligand
BDBM50108164
(CHEMBL308264 | N-[2-(4'-Cyano-biphenyl-4-sulfonyl)...)
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Affinity Data
IC50: 0.340nM
Assay Description:
In vitro selective inhibition against matrix metalloprotease-2 (MMP-2) using fluorimetric assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Interstitial collagenase
(Homo sapiens (Human))
Abbott Laboratories
Curated by
ChEMBL
Ligand
BDBM50108164
(CHEMBL308264 | N-[2-(4'-Cyano-biphenyl-4-sulfonyl)...)
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Copy InChI
Affinity Data
IC50: 3.60nM
Assay Description:
In vitro selective inhibition against matrix metalloprotease-1 (MMP-1) using a fluorimetric assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Matrix metalloproteinase-9
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50108164
(CHEMBL308264 | N-[2-(4'-Cyano-biphenyl-4-sulfonyl)...)
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Copy InChI
Affinity Data
IC50: 4.10nM
Assay Description:
Inhibition of MMP9
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Matrix metalloproteinase-9
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50108164
(CHEMBL308264 | N-[2-(4'-Cyano-biphenyl-4-sulfonyl)...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.10nM
Assay Description:
In vitro selective inhibition against Matrix metalloprotease-9 (MMP-9) using fluorimetric assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI