Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
MAP kinase-interacting serine/threonine-protein kinase 2
(Homo sapiens (Human))
Effector Therapeutics
US Patent
Ligand
BDBM297366
(7-chloro-3,3-dimethyl-5-(pyrimidin-4-ylamino)isoin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: <10nM
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
MAP kinase-interacting serine/threonine-protein kinase 1
(Homo sapiens (Human))
Effector Therapeutics
US Patent
Ligand
BDBM297366
(7-chloro-3,3-dimethyl-5-(pyrimidin-4-ylamino)isoin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: <10nM
Assay Description:
Compounds are screened for MNK inhibition using the ADP-Glo kinase assay kit (Promega, catalogue No. V9101). All kinase reactions are performed in Re...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI