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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Delta-type opioid receptor
(Homo sapiens (Human))
University Of Michigan
Curated by
ChEMBL
Ligand
BDBM50000653
(10-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
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Affinity Data
Ki: 26nM
Assay Description:
Compound was tested for the inhibition of [3H]- [D-Pen2, D-Pen5]-enkephalin (DPDPE) binding to Opioid receptor delta 1 in guinea pig brain homogenate...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Mu-type opioid receptor
(GUINEA PIG)
University Of Michigan
Curated by
ChEMBL
Ligand
BDBM50000653
(10-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
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Affinity Data
Ki: 3.45E+3nM
Assay Description:
Compound was tested for the inhibition of [3H]- [D-Ala2, N-MePhe4, Gly5-ol]-enkephalin (DAMGO) binding to Opioid receptor mu 1 in guinea pig brain ho...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Kappa-type opioid receptor
(Cavia porcellus (domestic guinea pig))
University Of Michigan
Curated by
ChEMBL
Ligand
BDBM50000653
(10-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
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Copy InChI
Affinity Data
Ki: >1.00E+4nM
Assay Description:
Compound was tested for the inhibition of [3H]- (U69,593) binding to Opioid receptor kappa 1 in guinea pig brain homogenates
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI