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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50041371((S)-10,13-Dimethyl-6-vinyl-1,6,7,8,9,10,11,12,13,1...)
Affinity DataKi:  5.10nMAssay Description:Binding affinity for human placental microsome aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50136064(CHEMBL3753920)
Affinity DataKi:  5.10nMAssay Description:Competitive inhibition of human aromatase extracted from placental microsomes after 10 mins in presence of [1beta-3H]androstenedioneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50041371((S)-10,13-Dimethyl-6-vinyl-1,6,7,8,9,10,11,12,13,1...)
Affinity DataIC50:  320nMAssay Description:Inhibitory concentration was tested on Cytochrome P450 19A1 in human placental microsomes 20 (microg) of protein incubated for 20 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed