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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50039155(13-Methyl-7,17-dioxo-1,2,7,8,9,11,12,13,14,15,16,1...)
Affinity DataKi:  1.80E+3nMAssay Description:The binding affinity was determined on Cytochrome P450 19A1 by analysis of Dixon plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50039155(13-Methyl-7,17-dioxo-1,2,7,8,9,11,12,13,14,15,16,1...)
Affinity DataKi:  2.90E+3nMAssay Description:Time dependent inactivation of aromatase cytochrome P450 19A1 from Kitz-Wilson plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Tohoku College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50039155(13-Methyl-7,17-dioxo-1,2,7,8,9,11,12,13,14,15,16,1...)
Affinity DataIC50:  1.10E+4nMAssay Description:In vitro competetitive inhibitory activity was measured on Cytochrome P450 19A1 of human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed