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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
13
hits in this display
Target
Induced myeloid leukemia cell differentiation protein Mcl-1
(Homo sapiens (Human))
Emory University
Curated by
PubChem BioAssay
Ligand
BDBM50269745
(CHEMBL463175 | Cephalochromin | cid_160115)
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Affinity Data
IC50: 1.49E+3nM
Assay Description:
NIH Molecular Libraries Screening Centers Network [MLSCN] Emory Chemical Biology Discovery Center in MLSCN Assay provider: Nikolovska-Coleska, Univer...
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Target Info
PDB
MMDB
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KEGG
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antibodypedia
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Target
Enoyl-[acyl-carrier-protein] reductase [NADH] FabI
(Escherichia coli)
TBA
Ligand
BDBM50269745
(CHEMBL463175 | Cephalochromin | cid_160115)
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Affinity Data
IC50: 1.80E+3nM
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Target
Enoyl-[acyl-carrier-protein] reductase [NADPH] FabI
(Staphylococcus aureus)
TBA
Ligand
BDBM50269745
(CHEMBL463175 | Cephalochromin | cid_160115)
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Affinity Data
IC50: 1.90E+3nM
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Target
Glucagon receptor
(Homo sapiens (Human))
Boehringer Ingelheim Pharma Gmbh And
Curated by
ChEMBL
Ligand
BDBM50269745
(CHEMBL463175 | Cephalochromin | cid_160115)
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Affinity Data
IC50: 2.00E+4nM
Assay Description:
Antagonist activity at human glucagon receptor expressed in BHK21 cells assessed as inhibition of glucagon-induced cAMP elevation by RIA
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Target Info
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Article
PubMed
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Target
Botulinum neurotoxin type A
(Clostridium botulinum (strain Hall / ATCC 3502 / N...)
TBA
Curated by
ChEMBL
Ligand
BDBM50269745
(CHEMBL463175 | Cephalochromin | cid_160115)
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Affinity Data
IC50: 2.92E+4nM
Assay Description:
Inhibition of Clostridium botulinum Hall BoNT/A protease activity using Ac-SNKTRIDEANQRATKML-NH2 as substrate after 5 mins by RP-HPLC analysis
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Target
Transitional endoplasmic reticulum ATPase
(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center
Curated by
PubChem BioAssay
Ligand
BDBM50269745
(CHEMBL463175 | Cephalochromin | cid_160115)
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Affinity Data
IC50: 4.39E+4nM
Assay Description:
Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...
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Target Info
PDB
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Target
Transitional endoplasmic reticulum ATPase
(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center
Curated by
PubChem BioAssay
Ligand
BDBM50269745
(CHEMBL463175 | Cephalochromin | cid_160115)
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Affinity Data
IC50: >5.00E+4nM
Assay Description:
Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...
More data for this Ligand-Target Pair
Target Info
PDB
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Target
M1 family aminopeptidase
(Plasmodium falciparum (isolate FcB1 / Columbia))
Srmlsc
Curated by
PubChem BioAssay
Ligand
BDBM50269745
(CHEMBL463175 | Cephalochromin | cid_160115)
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Affinity Data
IC50: 6.49E+4nM
Assay Description:
Southern Research Molecular Libraries Screening Center (SRMLSC) Southern Research Institute (Birmingham, Alabama) NIH Molecular Libraries Screening...
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Target
Intestinal-type alkaline phosphatase 1
(Rattus norvegicus (Rat))
Burnham Center For Chemical Genomics
Curated by
PubChem BioAssay
Ligand
BDBM50269745
(CHEMBL463175 | Cephalochromin | cid_160115)
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Affinity Data
EC50: 1.91E+4nM
Assay Description:
Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...
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Target Info
PDB
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Target
Alkaline phosphatase, tissue-nonspecific isozyme
(Homo sapiens (Human))
Burnham Center For Chemical Genomics
Curated by
PubChem BioAssay
Ligand
BDBM50269745
(CHEMBL463175 | Cephalochromin | cid_160115)
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Affinity Data
EC50: 2.67E+4nM
Assay Description:
Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...
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Target Info
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Target
Intestinal-type alkaline phosphatase
(Homo sapiens (Human))
Burnham Center For Chemical Genomics
Curated by
PubChem BioAssay
Ligand
BDBM50269745
(CHEMBL463175 | Cephalochromin | cid_160115)
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Affinity Data
EC50: 2.17E+4nM
Assay Description:
Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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KEGG
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Target
Streptokinase A
(Streptococcus pyogenes M1 GAS)
Broad Institute
Curated by
PubChem BioAssay
Ligand
BDBM50269745
(CHEMBL463175 | Cephalochromin | cid_160115)
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Affinity Data
EC50: 1.50E+5nM
Assay Description:
Keywords: Group A streptococcus, GAS, streptokinase, expression, virulence, inhibition, dose response, EC50 Assay Overview: The goal of this assa...
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Target
Alkaline phosphatase, germ cell type
(Homo sapiens (Human))
Burnham Center For Chemical Genomics
Curated by
PubChem BioAssay
Ligand
BDBM50269745
(CHEMBL463175 | Cephalochromin | cid_160115)
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Affinity Data
EC50: 2.11E+4nM
Assay Description:
Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
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