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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
ATP-sensitive inward rectifier potassium channel 1
(Homo sapiens (Human))
Merck Sharp & Dohme
US Patent
Ligand
BDBM194980
(US9206198, 39 | US9206198, 42)
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Affinity Data
IC50: 20nM
T: 2°C
Assay Description:
The ROMK channel functional thallium flux assay is performed in 384 wells, using the FLIPR-Tetra instrument. HEK-hKir1.1 cells are seeded in Poly-D...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
ATP-sensitive inward rectifier potassium channel 1
(Homo sapiens (Human))
Merck Sharp & Dohme
US Patent
Ligand
BDBM194980
(US9206198, 39 | US9206198, 42)
Copy SMILES
Copy InChI
Affinity Data
IC50: 100nM
T: 2°C
Assay Description:
The ROMK channel functional thallium flux assay is performed in 384 wells, using the FLIPR-Tetra instrument. HEK-hKir1.1 cells are seeded in Poly-D...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI