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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Guanine nucleotide-binding protein subunit alpha-15 [Y147C]/Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Merck Sharp & Dohme
US Patent
Ligand
BDBM212880
(US9278960, 2-27 | US9663506, Example 2-27)
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Affinity Data
IC50: 7nM
Assay Description:
The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Merck Sharp & Dohme
US Patent
Ligand
BDBM212880
(US9278960, 2-27 | US9663506, Example 2-27)
Copy SMILES
Copy InChI
Affinity Data
IC50: 7nM
Assay Description:
The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Merck Sharp & Dohme
US Patent
Ligand
BDBM212880
(US9278960, 2-27 | US9663506, Example 2-27)
Copy SMILES
Copy InChI
Affinity Data
IC50: 7nM
Assay Description:
The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI