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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
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Target
Transient receptor potential cation channel subfamily V member 1
(Homo sapiens (Human))
Sapienza University Of Rome
Curated by
ChEMBL
Ligand
BDBM50424152
(CHEMBL2312056)
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Affinity Data
IC50: 310nM
Assay Description:
Antagonist activity at human TRPV1 overexpressed in HEK293 cells assessed as inhibition of capsaicin-induced intracellular Ca2+ level incubated for 5...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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In Depth
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Article
PubMed
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Target
Transient receptor potential cation channel subfamily A member 1
(Rattus norvegicus)
Sapienza University Of Rome
Curated by
ChEMBL
Ligand
BDBM50424152
(CHEMBL2312056)
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Affinity Data
IC50: 3.51E+4nM
Assay Description:
Antagonist activity at rat TRPA1 overexpressed in HEK293 cells assessed as inhibition of allyl isothiocyanate-induced intracellular Ca2+ level incuba...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Sapienza University Of Rome
Curated by
ChEMBL
Ligand
BDBM50424152
(CHEMBL2312056)
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Affinity Data
IC50: >5.00E+4nM
Assay Description:
Inhibition of FAAH in rat brain homogenates using [14C]anandamide as substrate assessed as formation of [14C]ethanolamine after 30 mins by scintillat...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Transient receptor potential cation channel subfamily A member 1
(Rattus norvegicus)
Sapienza University Of Rome
Curated by
ChEMBL
Ligand
BDBM50424152
(CHEMBL2312056)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1.38E+4nM
Assay Description:
Agonist activity at rat TRPA1 overexpressed in HEK293 cells assessed as increase in allyl isothiocyanate-induced intracellular Ca2+ level by Fluo-4 b...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Transient receptor potential cation channel subfamily V member 1
(Homo sapiens (Human))
Sapienza University Of Rome
Curated by
ChEMBL
Ligand
BDBM50424152
(CHEMBL2312056)
Copy SMILES
Copy InChI
Affinity Data
EC50: 470nM
Assay Description:
Agonist activity at human TRPV1 overexpressed in HEK293 cells assessed as increase in ionomycin-induced intracellular Ca2+ level by Fluo-4 based spec...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI