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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMelatonin receptor type 1B(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50093292(CHEMBL133001 | N-Acenaphthen-1-ylmethyl-propionami...)
Affinity DataKi:  0.220nMAssay Description:Binding affinity for melatonin receptor type 1B, expressed in HEK-293 cells (2-[125I]-Iodomelatonin is used as radioligand)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50093292(CHEMBL133001 | N-Acenaphthen-1-ylmethyl-propionami...)
Affinity DataKi:  2.65nMAssay Description:Binding affinity for human melatonin receptor type 1A, expressed in HEK-293 cells (2-[125I]-Iodomelatonin is used as radioligand)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed