Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetAndrogen receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

LigandBDBM18562(6-alkyl, 7-amino-2-quinolinone, 11d (+/-) | 7-amin...)Copy SMILESCopy InChI

Affinity DataKi:  13nM IC50:  14nM EC50:  65nMAssay Description:The compounds were evaluated in a transcriptional activation assay with hAR in a mammalian cell background (CV-1) as the primary in vitro assay. Rece...More data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
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Ligand InfoPC cidPC sidSimilars

In DepthDetails ArticlePubMed
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