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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetLethal factor(Bacillus anthracis)
Panthera Biopharma

Curated by ChEMBL
LigandPNGBDBM50379534(CHEMBL2012837)
Affinity DataKi:  1nMAssay Description:Inhibition of N-terminal 6-histine tagged Bacillus anthracis LF 263-C terminal catalytic domain using MCA-KKVYPYPME-Dap(Dnp)-NH2 as substrate after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
Panthera Biopharma

Curated by ChEMBL
LigandPNGBDBM50379534(CHEMBL2012837)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of MMP-12 using OmniMMP as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Panthera Biopharma

Curated by ChEMBL
LigandPNGBDBM50379534(CHEMBL2012837)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of MMP-9 using OmniMMP as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Panthera Biopharma

Curated by ChEMBL
LigandPNGBDBM50379534(CHEMBL2012837)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of MMP-1 using OmniMMP as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Panthera Biopharma

Curated by ChEMBL
LigandPNGBDBM50379534(CHEMBL2012837)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of MMP-14 using OmniMMP as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Panthera Biopharma

Curated by ChEMBL
LigandPNGBDBM50379534(CHEMBL2012837)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of MMP-3 using OmniMMP as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Panthera Biopharma

Curated by ChEMBL
LigandPNGBDBM50379534(CHEMBL2012837)
Affinity DataIC50:  340nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Panthera Biopharma

Curated by ChEMBL
LigandPNGBDBM50379534(CHEMBL2012837)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of human ERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed