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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
9
hits in this display
Target
Neuropeptide Y receptor type 4
(Homo sapiens (Human))
University Of Cincinnati
Curated by
ChEMBL
Ligand
BDBM50185366
(CHEMBL2371911 | CHEMBL436499 | Sub[-Trp-Arg-Nva-Ar...)
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Affinity Data
Ki: 2nM
Assay Description:
Reduced farnesylation of H-ras transformed NIH3T3 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Neuropeptide Y receptor type 4
(Homo sapiens (Human))
University Of Cincinnati
Curated by
ChEMBL
Ligand
BDBM50185366
(CHEMBL2371911 | CHEMBL436499 | Sub[-Trp-Arg-Nva-Ar...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 2nM
Assay Description:
Inhibition of [3H]-FPP incorporation into biotin-linked K-ras decapeptide (CVIM) by bovine farnesyltransferase
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Neuropeptide Y receptor type 1
(Homo sapiens (Human))
University Of Cincinnati
Curated by
ChEMBL
Ligand
BDBM50185366
(CHEMBL2371911 | CHEMBL436499 | Sub[-Trp-Arg-Nva-Ar...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 80nM
Assay Description:
In vitro inhibitory activity against Factor Xa
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Neuropeptide Y receptor type 1
(Homo sapiens (Human))
University Of Cincinnati
Curated by
ChEMBL
Ligand
BDBM50185366
(CHEMBL2371911 | CHEMBL436499 | Sub[-Trp-Arg-Nva-Ar...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 80nM
Assay Description:
In vitro inhibitory activity against Factor Xa
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Neuropeptide Y receptor type 2
(Homo sapiens (Human))
University Of Cincinnati
Curated by
ChEMBL
Ligand
BDBM50185366
(CHEMBL2371911 | CHEMBL436499 | Sub[-Trp-Arg-Nva-Ar...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 390nM
Assay Description:
Displacement of [125I]NPY from human NPY2 receptor expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Neuropeptide Y receptor type 2
(Homo sapiens (Human))
University Of Cincinnati
Curated by
ChEMBL
Ligand
BDBM50185366
(CHEMBL2371911 | CHEMBL436499 | Sub[-Trp-Arg-Nva-Ar...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 530nM
Assay Description:
In vitro inhibitory activity against Factor Xa
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Neuropeptide Y receptor type 4
(Homo sapiens (Human))
University Of Cincinnati
Curated by
ChEMBL
Ligand
BDBM50185366
(CHEMBL2371911 | CHEMBL436499 | Sub[-Trp-Arg-Nva-Ar...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 430nM
Assay Description:
Agonist activity at human NPY4 receptor in HEK293 cells by inhibition of forskolin-stimulated cAMP synthesis
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Neuropeptide Y receptor type 1
(Homo sapiens (Human))
University Of Cincinnati
Curated by
ChEMBL
Ligand
BDBM50185366
(CHEMBL2371911 | CHEMBL436499 | Sub[-Trp-Arg-Nva-Ar...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1.41E+3nM
Assay Description:
Agonist activity at human NPY1 receptor in CHO cells by inhibition of forskolin-stimulated cAMP synthesis
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Neuropeptide Y receptor type 4
(Homo sapiens (Human))
University Of Cincinnati
Curated by
ChEMBL
Ligand
BDBM50185366
(CHEMBL2371911 | CHEMBL436499 | Sub[-Trp-Arg-Nva-Ar...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 370nM
Assay Description:
Inhibition of [3H]-FPP incorporation into biotin-linked K-ras decapeptide (CVIM) by bovine farnesyltransferase
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI