Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50333551(2-ethyl-5-(N-methyl-piperazin-1-yl)-1-(naphthalene...)
Affinity DataIC50:  4nMAssay Description:Displacement of [3H]mesulergine from human 5HT2C receptor expressed in cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50333551(2-ethyl-5-(N-methyl-piperazin-1-yl)-1-(naphthalene...)
Affinity DataIC50:  9nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50333551(2-ethyl-5-(N-methyl-piperazin-1-yl)-1-(naphthalene...)
Affinity DataIC50:  455nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50333551(2-ethyl-5-(N-methyl-piperazin-1-yl)-1-(naphthalene...)
Affinity DataIC50:  623nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50333551(2-ethyl-5-(N-methyl-piperazin-1-yl)-1-(naphthalene...)
Affinity DataIC50:  999nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50333551(2-ethyl-5-(N-methyl-piperazin-1-yl)-1-(naphthalene...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]spiperone from human dopamine D2 receptor expressed in cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50333551(2-ethyl-5-(N-methyl-piperazin-1-yl)-1-(naphthalene...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]spiperone from human dopamine D4 receptor expressed in cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50333551(2-ethyl-5-(N-methyl-piperazin-1-yl)-1-(naphthalene...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]LSD from human 5HT7 receptor expressed in cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed