Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetDelta-type opioid receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50306300(4-(4-(3-hydroxyphenyl)-1-(2-methylpentyl)piperidin...)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]diprenorphine from human delta opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50306300(4-(4-(3-hydroxyphenyl)-1-(2-methylpentyl)piperidin...)
Affinity DataKi:  150nMAssay Description:Displacement of [125I]diprenorphine from human kappa opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50306300(4-(4-(3-hydroxyphenyl)-1-(2-methylpentyl)piperidin...)
Affinity DataKi: >890nMAssay Description:Displacement of [125I]diprenorphine from human mu opioid receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50306300(4-(4-(3-hydroxyphenyl)-1-(2-methylpentyl)piperidin...)
Affinity DataIC50:  72nMAssay Description:Antagonist activity at delta opioid receptor by GTPgammaS bunding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed