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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Leucyl-cystinyl aminopeptidase
(Rattus norvegicus)
Astellas Pharma
US Patent
Ligand
BDBM271289
(US10059720, Example 104 | US10975091, Example 104)
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Copy InChI
Affinity Data
IC50: 21nM
Assay Description:
IRAP: Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP....
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Leucyl-cystinyl aminopeptidase
(Rattus norvegicus)
Astellas Pharma
US Patent
Ligand
BDBM271289
(US10059720, Example 104 | US10975091, Example 104)
Copy SMILES
Copy InChI
Affinity Data
IC50: 21nM
Assay Description:
Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Leucyl-cystinyl aminopeptidase
(Homo sapiens (Human))
Astellas Pharma
US Patent
Ligand
BDBM271289
(US10059720, Example 104 | US10975091, Example 104)
Copy SMILES
Copy InChI
Affinity Data
IC50: 26nM
Assay Description:
hP-LAP: HEK293 cells forced to transiently express hP-LAP were prepared by lipofection, homogenized, and then subjected to ultracentrifugation at 100...
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Leucyl-cystinyl aminopeptidase
(Homo sapiens (Human))
Astellas Pharma
US Patent
Ligand
BDBM271289
(US10059720, Example 104 | US10975091, Example 104)
Copy SMILES
Copy InChI
Affinity Data
IC50: 26nM
Assay Description:
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI