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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
8
hits in this display
Target
Melanocortin receptor 3
(Homo sapiens (Human))
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50184364
(CHEMBL203602 | c[Nle-Gln-D-Phe-Arg-Trp-Glu]-NH2)
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Affinity Data
IC50: 270nM
Assay Description:
Inhibitory activity against hMC3R transfected in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 5
(Homo sapiens (Human))
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50184364
(CHEMBL203602 | c[Nle-Gln-D-Phe-Arg-Trp-Glu]-NH2)
Copy SMILES
Copy InChI
Affinity Data
IC50: 500nM
Assay Description:
Inhibitory activity against hMC5R transfected in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocyte-stimulating hormone receptor
(Homo sapiens (Human))
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50184364
(CHEMBL203602 | c[Nle-Gln-D-Phe-Arg-Trp-Glu]-NH2)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.00E+3nM
Assay Description:
Inhibitory activity against hMC1R transfected in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 4
(Homo sapiens (Human))
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50184364
(CHEMBL203602 | c[Nle-Gln-D-Phe-Arg-Trp-Glu]-NH2)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibitory activity against hMC4R transfected in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 3
(Homo sapiens (Human))
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50184364
(CHEMBL203602 | c[Nle-Gln-D-Phe-Arg-Trp-Glu]-NH2)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1.70E+3nM
Assay Description:
Activity against hMC3R transfected in HEK293 cells by intracellular cAMP accumulation
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 5
(Homo sapiens (Human))
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50184364
(CHEMBL203602 | c[Nle-Gln-D-Phe-Arg-Trp-Glu]-NH2)
Copy SMILES
Copy InChI
Affinity Data
EC50: 300nM
Assay Description:
Activity against hMC5R transfected in HEK293 cells by intracellular cAMP accumulation
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 4
(Homo sapiens (Human))
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50184364
(CHEMBL203602 | c[Nle-Gln-D-Phe-Arg-Trp-Glu]-NH2)
Copy SMILES
Copy InChI
Affinity Data
EC50: >1.00E+4nM
Assay Description:
Activity against hMC4R transfected in HEK293 cells by intracellular cAMP accumulation
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocyte-stimulating hormone receptor
(Homo sapiens (Human))
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50184364
(CHEMBL203602 | c[Nle-Gln-D-Phe-Arg-Trp-Glu]-NH2)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1.00E+3nM
Assay Description:
Activity against hMC1R transfected in HEK293 cells by intracellular cAMP accumulation
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI