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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetMelanocortin receptor 5(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50184362(CHEMBL380638 | c[Nle-Nle-D-Phe-Arg-Trp-Glu]-NH2)
Affinity DataIC50:  70nMAssay Description:Inhibitory activity against hMC5R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50184362(CHEMBL380638 | c[Nle-Nle-D-Phe-Arg-Trp-Glu]-NH2)
Affinity DataIC50:  250nMAssay Description:Inhibitory activity against hMC3R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50184362(CHEMBL380638 | c[Nle-Nle-D-Phe-Arg-Trp-Glu]-NH2)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity against hMC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50184362(CHEMBL380638 | c[Nle-Nle-D-Phe-Arg-Trp-Glu]-NH2)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against hMC1R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50184362(CHEMBL380638 | c[Nle-Nle-D-Phe-Arg-Trp-Glu]-NH2)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity against hMC4R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50184362(CHEMBL380638 | c[Nle-Nle-D-Phe-Arg-Trp-Glu]-NH2)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity against hMC5R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50184362(CHEMBL380638 | c[Nle-Nle-D-Phe-Arg-Trp-Glu]-NH2)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity against hMC1R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50184362(CHEMBL380638 | c[Nle-Nle-D-Phe-Arg-Trp-Glu]-NH2)
Affinity DataEC50:  300nMAssay Description:Activity against hMC3R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed