Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50183555(CHEMBL408832 | H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-N...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50183555(CHEMBL408832 | H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-N...)
Affinity DataKi:  88nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50183555(CHEMBL408832 | H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-N...)
Affinity DataKi:  560nMAssay Description:Displacement of [125I]CCK8 from human CCK2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50183555(CHEMBL408832 | H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-N...)
Affinity DataKi:  560nMAssay Description:Displacement of [125I]CCK8 from human CCK2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50183555(CHEMBL408832 | H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-N...)
Affinity DataKi:  840nMAssay Description:Displacement of [125I]CCK8 from human CCK1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50183555(CHEMBL408832 | H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-N...)
Affinity DataKi:  840nMAssay Description:Displacement of [125I]CCK8 from human CCK1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50183555(CHEMBL408832 | H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-N...)
Affinity DataIC50:  38nMAssay Description:Agonist activity at delta opioid receptor by inhibition of muscle contraction in electrically stimulated isolated mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50183555(CHEMBL408832 | H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-N...)
Affinity DataIC50:  640nMAssay Description:Agonist activity at mu opioid receptor by inhibition of muscle contraction in electrically stimulated isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50183555(CHEMBL408832 | H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-N...)
Affinity DataEC50:  28nMAssay Description:Inhibition of [35S]GTP-gamma-S binding to human delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50183555(CHEMBL408832 | H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-N...)
Affinity DataEC50:  10nMAssay Description:Inhibition of [35S]GTP-gamma-S binding to rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50183555(CHEMBL408832 | H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-N...)
Affinity DataEC50:  10nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed