Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM250634(US9447148, 9.2 | US9447148, 9.31)
BDBM250634(US9447148, 9.2 | US9447148, 9.31)
Ki: 2nM ΔG°: -51.6kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMCR-1a or hMCR-...More data for this Ligand-Target Pair
BDBM250634(US9447148, 9.2 | US9447148, 9.31)
Ki: 110nM ΔG°: -41.3kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMCR-1a or hMCR-...More data for this Ligand-Target Pair
BDBM250634(US9447148, 9.2 | US9447148, 9.31)
Ki: 1.00E+4nM ΔG°: -29.7kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMCR-1a or hMCR-...More data for this Ligand-Target Pair
BDBM250634(US9447148, 9.2 | US9447148, 9.31)
BDBM250634(US9447148, 9.2 | US9447148, 9.31)
EC50: 0.00600nMpH: 7.5 T: 2°CAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair