Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM250639(US9447148, 9.7)
Affinity DataKi:  0.550nM ΔG°:  -55.0kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMCR-1a or hMCR-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM250639(US9447148, 9.7)
Affinity DataKi:  33nM ΔG°:  -44.4kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMCR-1a or hMCR-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM250639(US9447148, 9.7)
Affinity DataEC50:  0.0250nMpH: 7.5 T: 2°CAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent