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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156358(2-Hydroxymethyl-6-propyl-piperidine-3,4,5-triol | ...)
Affinity DataIC50:  530nMAssay Description:Inhibition of rat intestinal isomaltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative alpha-glucosidase(Oryza sativa subsp. japonica)
Universit£

Curated by ChEMBL
LigandPNGBDBM50156358(2-Hydroxymethyl-6-propyl-piperidine-3,4,5-triol | ...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibitory activity against alpha-Glucosidase from riceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156358(2-Hydroxymethyl-6-propyl-piperidine-3,4,5-triol | ...)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of rat intestinal sucrase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156358(2-Hydroxymethyl-6-propyl-piperidine-3,4,5-triol | ...)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of rat intestinal maltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
Hokuriku University

LigandPNGBDBM18360((2R,3R,4R,5S,6R)-2-(hydroxymethyl)-6-propylpiperid...)
Affinity DataIC50:  2.70E+5nMpH: 4.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Hokuriku University

LigandPNGBDBM18360((2R,3R,4R,5S,6R)-2-(hydroxymethyl)-6-propylpiperid...)
Affinity DataIC50:  4.00E+5nMpH: 5.5 T: 2°CAssay Description:Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Hokuriku University

LigandPNGBDBM18360((2R,3R,4R,5S,6R)-2-(hydroxymethyl)-6-propylpiperid...)
Affinity DataIC50:  4.00E+5nMAssay Description:Inhibition of human recombinant beta-glucocerebrosidase preincubated for 10 mins before 4-methylumbelliferyl-betaD-glucopyranoside addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Hokuriku University

LigandPNGBDBM50315251((2S,3R,4R,5S,6S)-2-(hydroxymethyl)-6-propylpiperid...)
Affinity DataIC50:  4.87E+5nMAssay Description:Inhibition of human recombinant beta-glucocerebrosidase assessed as p-nitrophenolate accumulation preincubated for 10 mins before p-nitrophenyl-beta-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50437449(CHEMBL2409342)
Affinity DataIC50:  7.13E+5nMAssay Description:Inhibition of bovine kidney alpha-L-fucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed