Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126094(CHEMBL437822 | MT-II cyclic peptide derivative)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126094(CHEMBL437822 | MT-II cyclic peptide derivative)
Affinity DataEC50:  1.33E+3nMAssay Description:Agonist activity at human melanocortin receptor (hMC1R).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed