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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50204382(2-(benzyloxyamino)-N-hydroxyhexanamide | CHEMBL228...)
Affinity DataKi:  7.60E+3nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 by CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50204382(2-(benzyloxyamino)-N-hydroxyhexanamide | CHEMBL228...)
Affinity DataKi:  7.80E+3nMAssay Description:Inhibition of human recombinant carbonic anhydrase 2 by CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50204382(2-(benzyloxyamino)-N-hydroxyhexanamide | CHEMBL228...)
Affinity DataKi:  5.20E+5nMAssay Description:Inhibition of human recombinant carbonic anhydrase 1 by CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50204382(2-(benzyloxyamino)-N-hydroxyhexanamide | CHEMBL228...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of Bacillus thermoproteolyticus pseudolysin pretreated with compound for 15 mins followed by the addition of Abz-Ala-Gly-leu-Ala-p-nitrobe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50204382(2-(benzyloxyamino)-N-hydroxyhexanamide | CHEMBL228...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa pseudolysin pretreated with compound for 1 hr followed by the addition of 1.73 uM bradykinin like substrate by s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50204382(2-(benzyloxyamino)-N-hydroxyhexanamide | CHEMBL228...)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of Bacillus thermoproteolyticus thermolysin pretreated with compound for 1 hr followed by the addition of 3.33 uM bradykinin like substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50204382(2-(benzyloxyamino)-N-hydroxyhexanamide | CHEMBL228...)
Affinity DataIC50:  3.37E+4nMAssay Description:Inhibition of human recombinant MMP2 expressed in mouse myeloma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50204382(2-(benzyloxyamino)-N-hydroxyhexanamide | CHEMBL228...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of recombinant human MMP2 after 2 hrs using FS-6 as substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50204382(2-(benzyloxyamino)-N-hydroxyhexanamide | CHEMBL228...)
Affinity DataIC50:  8.10E+4nMAssay Description:Inhibition of recombinant human MMP9 after 2 hrs using FS-6 as substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50204382(2-(benzyloxyamino)-N-hydroxyhexanamide | CHEMBL228...)
Affinity DataIC50:  8.15E+4nMAssay Description:Inhibition of human recombinant MMP9 expressed in mouse myeloma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Uit The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50204382(2-(benzyloxyamino)-N-hydroxyhexanamide | CHEMBL228...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of recombinant human ADAM17 after 30 mins using FS-6 as substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed