Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAdenosine receptor A1(Rattus norvegicus (rat))
Griffith University

Curated by ChEMBL

LigandBDBM50053941(2-(4-Amino-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-...)Copy SMILESCopy InChI

Affinity DataKi:  0.939nMAssay Description:Displacement of [3H]-N6-PIA from Adenosine A1 receptor from rat whole brainMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Griffith University

Curated by ChEMBL

LigandBDBM50053941(2-(4-Amino-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-6-...)Copy SMILESCopy InChI

Affinity DataKi:  88.3nMAssay Description:Inhibition of [3H]-CGS-21,680 binding to Adenosine A2A receptor of rat striatal membranesMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI