Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMelanocortin receptor 4(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50220690((R)-N-((S)-1-(4-butyl-4-(cyanomethyl)piperidin-1-y...)
Affinity DataIC50:  22nMAssay Description:Binding affinity to human MC4RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50220690((R)-N-((S)-1-(4-butyl-4-(cyanomethyl)piperidin-1-y...)
Affinity DataEC50:  281nMAssay Description:Antagonist activity at human MC4R assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50220690((R)-N-((S)-1-(4-butyl-4-(cyanomethyl)piperidin-1-y...)
Affinity DataEC50:  480nMAssay Description:Antagonist activity at human MC5R assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed