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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50042226(4'-(2-Butyl-4-oxo-1,3-diaza-spiro[4.4]non-1-en-3-y...)
Affinity DataIC50:  269nMAssay Description:Inhibition of human serum AChE by Ellman colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50042226(4'-(2-Butyl-4-oxo-1,3-diaza-spiro[4.4]non-1-en-3-y...)
Affinity DataIC50:  271nMAssay Description:Inhibition of Wistar rat brain AChE by Ellman colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50042226(4'-(2-Butyl-4-oxo-1,3-diaza-spiro[4.4]non-1-en-3-y...)
Affinity DataIC50:  277nMAssay Description:Inhibition of electric eel AChE by Ellman colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Sanofi Recherche

Curated by ChEMBL
LigandPNGBDBM50042226(4'-(2-Butyl-4-oxo-1,3-diaza-spiro[4.4]non-1-en-3-y...)
Affinity DataIC50:  3.20E+3nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 measured by ability to displace [125I]- A II from its specific binding site in rat liver membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed