Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 5 hits in this display
BDBM50072714(5-Butyl-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza...)
Ki: 0.950nMAssay Description:Binding affinity was determined against hPR-A (human progesterone receptor) using progesterone radioligand in competitive binding assayMore data for this Ligand-Target Pair
BDBM50072714(5-Butyl-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza...)
BDBM50072714(5-Butyl-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza...)
BDBM50072714(5-Butyl-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza...)
BDBM50072714(5-Butyl-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza...)
EC50: 11nMAssay Description:Binding affinity was determined against hPR-A (human progesterone receptor) using progesterone radioligand in competitive binding assayMore data for this Ligand-Target Pair