Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetB2 bradykinin receptor(Cavia porcellus)
Fujisawa Pharmaceutical

Curated by ChEMBL

LigandBDBM50067252(CHEMBL338682 | Hexanoic acid ({[3-(3-bromo-2-methy...)Copy SMILESCopy InChI

Affinity DataIC50:  5.60nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair

Target InfoMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetB2 bradykinin receptor(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL

LigandBDBM50067252(CHEMBL338682 | Hexanoic acid ({[3-(3-bromo-2-methy...)Copy SMILESCopy InChI

Affinity DataIC50:  240nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI