Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetNociceptin receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50120140(C-{(R)-C-(3-Chloro-phenyl)-C-[(S)-1-(1-phenyl-hexy...)
Affinity DataKi:  34nMAssay Description:Binding affinity at human ORL1 receptor was determined by using [125I]nociceptin radioligand in Chinese hamster ovary (CHO) cell membranes at a conce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50120140(C-{(R)-C-(3-Chloro-phenyl)-C-[(S)-1-(1-phenyl-hexy...)
Affinity DataKi:  1.94E+3nMAssay Description:Binding affinity at human opioid receptor mu 1 was determined by using [3H]diprenorphine radioligand in CHO cell membranes at a concentration of 0.12...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50120140(C-{(R)-C-(3-Chloro-phenyl)-C-[(S)-1-(1-phenyl-hexy...)
Affinity DataKi:  2.99E+3nMAssay Description:Binding affinity at human opioid receptor kappa 1 was determined by using [3H]diprenorphine radioligand in CHO cell membranes at a concentration of 0...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50120140(C-{(R)-C-(3-Chloro-phenyl)-C-[(S)-1-(1-phenyl-hexy...)
Affinity DataKi:  5.96E+3nMAssay Description:Binding affinity at human opioid receptor delta 1 was determined by using [3H]diprenorphine radioligand in CHO cell membranes at a concentration of 0...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed