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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetStromelysin-1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50246795(CHEMBL509270 | N'-{3-(E)-[2-(S)-(2-Phenyl-1H-indol...)
Affinity DataIC50:  174nMAssay Description:Inhibition of human recombinant MMP3 catalytic domain by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50246795(CHEMBL509270 | N'-{3-(E)-[2-(S)-(2-Phenyl-1H-indol...)
Affinity DataIC50:  732nMAssay Description:Inhibition of human recombinant pro-MMP9 by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50246795(CHEMBL509270 | N'-{3-(E)-[2-(S)-(2-Phenyl-1H-indol...)
Affinity DataIC50:  1.27E+3nMAssay Description:Inhibition of human recombinant pro-MMP2 by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50246795(CHEMBL509270 | N'-{3-(E)-[2-(S)-(2-Phenyl-1H-indol...)
Affinity DataIC50:  2.04E+3nMAssay Description:Inhibition of human recombinant pro-MMP1 by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50246795(CHEMBL509270 | N'-{3-(E)-[2-(S)-(2-Phenyl-1H-indol...)
Affinity DataIC50:  3.78E+3nMAssay Description:Inhibition of human recombinant MMP14 catalytic domain by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed