Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetSerine/threonine-protein kinase B-raf [V600E](Homo sapiens (Human))
Beigene

US Patent

LigandBDBM200782(US9670231, 1.69)Copy SMILESCopy InChI

Affinity DataIC50:  2nMAssay Description:TBDMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoKEGGPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI

TargetEpidermal growth factor receptor [L858R](Homo sapiens (Human))
Beigene

US Patent

LigandBDBM200782(US9670231, 1.69)Copy SMILESCopy InChI

Affinity DataIC50:  116nMAssay Description:TBDMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoKEGGPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI

TargetEpidermal growth factor receptor(Homo sapiens (Human))
Beigene

US Patent

LigandBDBM200782(US9670231, 1.69)Copy SMILESCopy InChI

Affinity DataIC50:  118nMAssay Description:TBDMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoKEGGPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI

TargetEpidermal growth factor receptor [T790M,L858R](Homo sapiens (Human))
Beigene

US Patent

LigandBDBM200782(US9670231, 1.69)Copy SMILESCopy InChI

Affinity DataIC50:  782nMAssay Description:TBDMore data for this Ligand-Target Pair

Target InfoPDBMMDBKEGG
UniProtKB/SwissProt
B.MOADDrugBankGoogleScholar

Ligand InfoKEGGPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI