Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetStromelysin-1(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50070236(2-(2-Mercapto-acetyl)-nonanoic acid {(S)-2,2-dimet...)
Affinity DataIC50:  22nMAssay Description:In vitro inhibitory activity against stromelysin-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50070236(2-(2-Mercapto-acetyl)-nonanoic acid {(S)-2,2-dimet...)
Affinity DataIC50:  200nMAssay Description:In vitro inhibitory activity against collagenase-1(MMP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed